Adrenergic alpha-1 Receptor Antagonists: Products

α1 and α2B antagonist; also MT3 antagonist

Non-competitive NMDA antagonist; also σ ligand

α1 and α2B antagonist (α1 > α2B). Orally active

Highly selective α1 antagonist

α1A antagonist

Potent, subtype-selective α1A antagonist

Potent and non-selective β antagonist; also potent α1 antagonist

α1 antagonist

Selective α1A antagonist

5-HT2A and α1 adrenoceptor antagonist; also enhances neural differentiation; antidepressant and neuroprotectant

Adrenergic α receptor antagonist; antihypertensive

Selective α1A antagonist