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TRPV antagonist; also activator of ENaCδ
Potent and selective TRPV1 competitive antagonist
Non-selective CaV2.1 and 2.2 blocker; also blocks TRPV channels
Potent and selective TRPV4 antagonist
Potent and selective TRPV4 antagonist; orally active
Antiallergic; inhibits inflammatory mediator release from mast cells
Potent and selective TRPV1 competitive antagonist
Reversible, competitive and potent TRPV1 antagonist
Selective TRPV4 antagonist
Selective TRPV3 antagonist; brain penetrant
Potent and selective TRPV1 antagonist
Potent and selective TRPV1 antagonist
Potent and selective TRPV4 antagonist
Selective TRPV2 antagonist