Octreotide
Purity: ≥95%
Biological Activity
Octreotide is a peptide agonist for sst2, sst3 and sst5 somatostatin receptors. IC50/Kd values (nM) at cloned human somatostatin receptors are: 290 - 1140 (sst1), 0.4 - 2.1 (sst2), 4.4 - 34.5 (sst3), > 1000 (sst4), and 5.6 - 32 (sst5).Technical Data
(Modifications: Phe-1 = D-Phe, Trp-4 = D-Trp, Thr-8 = Thr-ol, Disulfide bridge between 2-7)
The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.
Background References
-
Molecular pharmacology of somatostatin receptors.
Hoyer et al.
Naunyn Schmiedebergs Arch.Pharmacol., 1994;350:441 -
Cloned somatostatin receptors: identification of subtype-selective peptides and demonstration of high affinity binding to linear peptides.
Raynor et al.
Mol.Pharmacol., 1993;43:838 -
Drug design at peptide receptors. Somatostatin receptor ligands.
Hannon et al.
J.Mol.Neurosci., 2002;18:15
Product Datasheets
Reconstitution Calculator
Molarity Calculator
FAQs
No product specific FAQs exist for this product, however you may
View all Peptide FAQsReviews for Octreotide
There are currently no reviews for this product. Be the first to review Octreotide and earn rewards!
Have you used Octreotide?
Submit a review and receive an Amazon gift card.
$25/€18/£15/$25CAN/¥75 Yuan/¥2500 Yen for a review with an image
$10/€7/£6/$10 CAD/¥70 Yuan/¥1110 Yen for a review without an image
