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AR-M 1000390 hydrochloride

Catalog #: 4335
3 Citations Datasheet / COA / SDS

Discontinued Product

4335 has been discontinued.
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AR-M 1000390 hydrochloride | CAS No. 209808-47-9 | delta Opioid Receptor Agonists
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Description: Low-internalizing δ agonist

Chemical Name: N,N-Diethyl-4-(phenyl-4-piperidinylidenemethyl)-benzamide hydrochloride

Purity: ≥97%

Product Details
Citations (3)
Reviews
Biological Activity Technical Data Background Product Datasheets Calculators

Biological Activity

AR-M 1000390 hydrochloride is a non-peptidic, low-internalizing δ-selective opioid receptor agonist; derivative of SNC 80 (Cat. No. 0764). Does not trigger acute desensitization of the analgesic response; reduces CFA-induced hyperalgesia. Brain penetrant following systemic administration.

Technical Data

M.Wt:
384.94
Formula:
C23H28N2O.HCl
Solubility:
Soluble to 100 mM in water and to 100 mM in DMSO
Purity:
≥97%
Storage:
Store at -20°C
CAS No:
209808-47-9

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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Citations for AR-M 1000390 hydrochloride

The citations listed below are publications that use Tocris products. Selected citations for AR-M 1000390 hydrochloride include:

3 Citations: Showing 1 - 3

  1. Subcellular location defines GPCR signal transduction.
    Authors: Francesco Luigi Et al.
    Sci Adv  2023;9:eadf6059
  2. Agonist-induced phosphorylation bar code and differential post-activation signaling of the delta opioid receptor revealed by phosphosite-specific antibodies.
    Authors: Anika Et al.
    Sci Rep  2020;10:8585
  3. A Genetically Encoded Biosensor Reveals Location Bias of Opioid Drug Action.
    Authors: Stoeber Et al.
    Neuron  2018;98:963

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