rac-CCT 250863

Catalog # Availability Size / Price Qty
4546/5
rac-CCT 250863 | CAS No. 1364269-06-6 | Nek2 Kinase Inhibitors
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Description: Potent Nek2 inhibitor

Chemical Name: 4-[2-Amino-5-[4-[(dimethylamino)methyl]-2-thienyl]-3-pyridinyl]-2-[[(2Z)-4,4,4-trifluoro-1-methyl-2-buten-1-yl]oxy]benzamide

Purity: ≥98%

Product Details
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Biological Activity

rac-CCT 250863 is a potent Nek2 inhibitor (IC50 = 73 nM). Exhibits selectivity for Nek2 over PLK1, MPS1, Cdk2 and Aurora A.

Technical Data

M.Wt:
490.54
Formula:
C24H25F3N4O2S
Solubility:
Soluble to 100 mM in 1eq. HCl and to 100 mM in DMSO
Purity:
≥98%
Storage:
Store at -20°C
CAS No:
1364269-06-6

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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