Home / Galanin Receptor Agonists / M617

M617

Catalog #: 2697
1 Citation Datasheet / COA / SDS
Catalog # Availability Size / Price Qty
2697/1
M617
1 Image
Description: Selective GAL1 agonist
Alternative Names: Galanin(1-13)-Gln14-bradykinin(2-9)amide

Purity: ≥95%

Product Details
Citations (1)
Supplemental Products
Reviews
Biological Activity Technical Data Background Product Datasheets Calculators

Biological Activity

M617 is a selective galanin GAL1 receptor agonist (Ki values are 0.23 and 5.71 nM for GAL1 and GAL2 receptors respectively). Enhances food consumption in rats following i.c.v. administration and reduces CAP-induced inflammatory pain.

Technical Data

M.Wt:
2361.68
Formula:
C112H161N29O28
Sequence:
GWTLNSAGYLLGPQPPGFSPFR

(Modifications: Arg-22 = C-terminal amide)

Solubility:
Soluble to 1 mg/ml in water
Purity:
≥95%
Storage:
Store at -20°C
CAS No:
860790-38-1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Background References

  1. Regulation of kindling epileptogenesis by hippocampal galanin type 1 and type 2 receptors: the effects of subtype-selective agonists and the role of G-protein-mediated signaling.
    Mazarati et al.
    J.Pharmacol.Exp.Ther., 2006;318:700
  2. Activation of peripheral galanin receptors: differential effects on nociception.
    Jimenez-Andrade et al.
    Pharmacol.Biochem.Behav., 2006;85:273
  3. A galanin receptor subtype 1 specific agonist.
    Lundstrom et al.
    Int.J.Pept.Res.Ther., 2005;11:17

Product Datasheets

COA view current batch
Or select another batch:
View Batch
SDS
Reconstitution Calculator
Molarity Calculator

Reconstitution Calculator

The reconstitution calculator allows you to quickly calculate the volume of a reagent to reconstitute your vial. Simply enter the mass of reagent and the target concentration and the calculator will determine the rest.

=
÷

Molarity Calculator

=
x
x
g/mol

*When preparing stock solutions always use the batch-specific molecular weight of the product found on the vial label and CoA (available online).

Citation for M617

The citations listed below are publications that use Tocris products. Selected citations for M617 include:

1 Citation: Showing 1 - 1

  1. Involvement of galanin and galanin receptor 1 in nociceptive modulation in the central nucleus of amygdala in normal and neuropathic rats.
    Authors: Li
    Sci Rep  2017;7(1):15317

FAQs

No product specific FAQs exist for this product, however you may

View all Peptide FAQs
Loading...

Reviews for M617

There are currently no reviews for this product. Be the first to review M617 and earn rewards!

Have you used M617?

Submit a review and receive an Amazon gift card.

$25/€18/£15/$25CAN/¥75 Yuan/¥1250 Yen for a review with an image

$10/€7/£6/$10 CAD/¥70 Yuan/¥1110 Yen for a review without an image

Submit a Review
Tocris Bioscience is the leading supplier of novel and exclusive tools for life science research with over 30 years' experience in the industry. Tocris is a Bio-Techne brand.