Home / Nicotinic (a7) Receptor Modulators / LY 2087101

LY 2087101

Catalog #: 4141
1 Citation Datasheet / COA / SDS
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4141/10
4141/50
LY 2087101 | CAS No. 913186-74-0 | Nicotinic (a7) Receptor Modulators
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Description: Allosteric potentiator of α7, α4β2 and α4β4 nAChRs

Chemical Name: [2-[(4-Fluorophenyl)amino]-4-methyl-5-thiazolyl]-3-thienylmethanone

Purity: ≥98%

Product Details
Citations (1)
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Biological Activity

LY 2087101 is an allosteric potentiator of α7, α4β2 and α4β4 nAChRs; displays selectivity against α3β4 nAChRs. Thought to potentiate agonist-evoked α7 responses by binding within the nAChR transmembrane region.

Technical Data

M.Wt:
318.39
Formula:
C15H11FN2OS2
Solubility:
Soluble to 100 mM in DMSO and to 10 mM in ethanol
Purity:
≥98%
Storage:
Store at +4°C
CAS No:
913186-74-0

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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Citation for LY 2087101

The citations listed below are publications that use Tocris products. Selected citations for LY 2087101 include:

1 Citation: Showing 1 - 1

  1. Studying Nicotinic Acetylcholine Receptors Using the IonFlux™ Microfluidic-Based Automated Patch-Clamp System with Continuous Perfusion and Fast Solution Exchange.
    Authors: Haiyang Et al.
    Curr Protoc Pharmacol  2020;88:e73

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