Home / KISS-Derived Peptide Receptor Antagonists / Kisspeptin 234

Kisspeptin 234

Catalog #: 3881
4 Citations Datasheet / COA / SDS
Catalog # Availability Size / Price Qty
3881/1
Kisspeptin 234
1 Image
Description: Kisspeptin receptor antagonist; kisspeptin 10 (Cat. No. 2570) analog

Purity: ≥95%

Product Details
Citations (4)
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Biological Activity

Kisspeptin 234 is a kisspeptin receptor (KISS1, GPR54) antagonist; kisspeptin-10 (Cat. No. 2570) analog. Inhibits kisspeptin-10 stimulation of inositol phosphate (IP) (IC50 = 7 nM) and release of gonadotrophin-releasing hormone (GnRH).

Technical Data

M.Wt:
1295.42
Formula:
C63H78N18O13
Sequence:
Ac-ANWNGFGWRF-NH2

(Modifications: Ala-1 = D-Ala & N-terminal Ac, Trp-8 = D-Trp, Phe-10 = C-terminal amide)

Solubility:
Soluble to 1 mg/ml in water
Purity:
≥95%
Storage:
Store at -20°C
CAS No:
1145998-81-7

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Additional Information

Licensing Caveats:
Sold under license

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Citations for Kisspeptin 234

The citations listed below are publications that use Tocris products. Selected citations for Kisspeptin 234 include:

4 Citations: Showing 1 - 4

  1. Kisspeptins inhibit human airway smooth muscle proliferation.
    Authors: Y S Et al.
    JCI Insight  2022;7
  2. Kisspeptin-54 attenuates oxidative stress and neuronal apoptosis in early brain injury after subarachnoid hemorrhage in rats via GPR54/ARRB2/AKT/GSK3β signaling pathway.
    Authors: Lei Et al.
    Free Radic Biol Med  2021;171:99-111
  3. The pregnant mouse uterus exhibits a functional kisspeptin/KISS1R signaling system on the day of embryo implantation.
    Authors: Fayazi Et al.
    Am J Physiol Renal Physiol  2015;13:105
  4. GPR54-dependent stimulation of luteinizing hormone secretion by neurokinin B in prepubertal rats.
    Authors: Grachev Et al.
    Reprod Biol Endocrinol  2012;7:e44344

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